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prasterone (Mylis)

✓ Approved

Merck & Co. · AR · Small Molecule

What is prasterone?

prasterone is a small molecule developed by Merck & Co.. It is approved for therapeutic indications.

Drug Profile

Brand NamesMylis
CompanyMerck & Co.
Drug ClassSmall Molecule
Molecular TargetAR
StatusApproved

Mechanism of Action

Molecular Targets

prasterone acts on 1 molecular target:

ARandrogen receptor (DHTR, AR8)
Want deeper analysis?Noah AI can explain complex mechanisms and compare to similar drugs.

Therapeutic Indications

prasterone is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Surgical and medical proceduresLabour induction✓ Approved

Related Research Articles

PubMedMobile DNA2026-07-16

Transposable element dynamics and regulatory role in sika deer (Cervus nippon) antler development.

Wang Qianghui Q, Xing Haihua H, Ma Yukai Y, Sun Zihui Z et al.

Deer antlers represent one of the few mammalian organs capable of complete regeneration, yet the underlying genomic regulatory mechanisms remain incompletely understood. Transposable elements (TEs), as key drivers of genome evolution and gene regulation, may play pivotal roles in the evolution of complex traits. This study aimed to systematically investigate the evolutionary dynamics of TEs in sika deer genome and to elucidate their potential regulatory functions in the development of antler by integrating comparative and functional genomics approaches. Comparative genomics revealed a lineage-specific massive expansion of LINE retrotransposons (dominated by RTE-BovB and L1 subfamilies) in cervid genomes, particularly in sika deer and red deer, where they constitute over 29% of the genomic sequence. The peak of this expansion (~ 7.5 million years ago) coincides with the major cladogenesis events within Cervus. Expression analysis showed that approximately 8.88% of annotated TEs are transcriptionally active in antler mesenchyme, with LINE and LTR elements being predominant among the 1,191 TEs consistently highly expressed across all stages. We identified numerous stage-specifically expressed TEs (SETEs) and found positive correlations between SETEs and key antler development genes, such as the osteogenic master regulator RUNX2, the extracellular matrix remodeling gene ANPEP, and the collagen synthesis gene P4HA3. Enrichment analysis demonstrated that genes adjacent to these TEs are significantly involved in pathways crucial for regeneration and rapid growth, including Wnt signaling, Hippo signaling, regulation of the actin cytoskeleton, and protein digestion and absorption. Our findings point to a potential role for cervid TEs expansion in driving genomic evolution and the acquisition of cervid-specific phenotypes, particularly antler growth and development. Through profiling TE expression in antler mesenchymal tissue across key development stages, the results suggest that dynamic TEs expression may be involved in the regulation of antler development, implicating a potential regulatory role for TEs in this rapid growth process. This study provides new insights into the molecular mechanisms underlying the rapid growth of antlers.

PubMedInternational journal of gynaecology and obstetrics: the official organ of the International Federation of Gynaecology and Obstetrics2026-07-15

Assessment and management of dyspareunia in peri- and postmenopausal women: A phenotype-based gynecologic approach.

Broul Marek M, Vančo Marcel M, Banýrová Jaroslava J, Hujová Aneta A

Dyspareunia in peri- and postmenopausal women is common, clinically consequential, and often undertreated in gynecologic practice. Although genitourinary syndrome of menopause (GSM) is a frequent contributor, intercourse-related pain may also reflect vestibular, pelvic floor, dermatologic, inflammatory, treatment-related, and psychosocial factors. This narrative review provides a practical phenotype-based framework for assessment and management when GSM, vestibular pain, and pelvic floor dysfunction coexist, and when deep-pain phenotypes require broader pelvic evaluation. PubMed/MEDLINE, the Cochrane Library, and selected guideline sources were searched for English-language literature published from January 2014 to March 2026, prioritizing guidelines, systematic reviews, randomized or sham-controlled trials, and examination-based studies relevant to office gynecology. History should distinguish superficial from deep pain, provoked from spontaneous symptoms, and urinary, dermatologic, inflammatory, and psychosocial features. Examination should proceed from vulva and vestibule to vagina and pelvic floor, with bimanual assessment and selective imaging when deeper pathology is suspected. Management includes education, irritant avoidance, moisturizers and lubricants, and prescription therapy for clinically significant GSM, usually low-dose vaginal estrogen, with prasterone or ospemifene as selected alternatives. Pelvic floor physiotherapy should be considered when tenderness, guarding, or penetration-limiting hypertonicity is present. Because menopause-specific pelvic floor evidence remains limited, related recommendations are framed as cautious extrapolations from broader dyspareunia, vulvodynia, and chronic pelvic pain literature.

PubMedInternational journal for parasitology. Parasites and wildlife2026-07-13

Phylogenetic and molecular insights into the genetic diversity of the invasive nematode Ashworthius sidemi infecting Poland's free-ranging European bison (Bison bonasus).

Świsłocka-Cutter Magdalena M, Borkowska Anetta A, Kowalczyk Rafał R, Kołodziej-Sobocińska Marta M

The invasive blood-sucking nematode Ashworthius sidemi, originally parasitising Asian cervids, has spread across Europe following human-mediated introductions of sika deer (Cervus nippon). In this study, we characterised the molecular variation of A. sidemi obtained from two neighbouring populations of European bison (Bison bonasus) in northeastern Poland, located in the Białowieża Primeval Forest and Knyszyńska Forest. Individual worms (one per host) were analysed using nuclear molecular markers (18S rRNA, 28S rRNA, ITS-1) and mitochondrial markers (COX1, ND4). All analysed markers revealed no detectable intraspecific genetic variability among the 16 specimens sequenced, with a single haplotype identified for each marker. This finding is consistent with a founder effect and/or recent introduction of the parasite. The genetic homogeneity observed across geographically close bison herds may also reflect host mobility. Phylogenetic analyses based on both nuclear and mitochondrial markers consistently placed A. sidemi within the subfamily Haemonchinae, closely related to Haemonchus spp. and Mecistocirrus digitatus. The ITS-1, COX1, and ND4 markers provided sufficient resolution to differentiate A. sidemi from other Trichostrongylidae species, whereas the 18S and 28S rRNA genes were too conserved to discriminate species- or subfamily-level relationships. Our findings demonstrate the utility of nuclear and mitochondrial markers for the identification and phylogenetic classification of trichostrongyloid nematodes. These results provide important insights into the invasion dynamics of A. sidemi, which may support parasite surveillance and conservation efforts of endangered host species.

PubMedAnimal science journal = Nihon chikusan Gakkaiho2026-07-11

Diversity of the Major Histocompatibility Complex Region Among Seven Founders of the Crested Ibis Nipponia nippon in Japan.

Taniguchi Yukio Y, Yamada Takahisa T, Sugiyama Toshie T, Kaneko Yoshinori Y et al.

The Crested Ibis Nipponia nippon is a critically threatened avian species. The current Japanese population originates from only seven founders introduced from China. The major histocompatibility complex (MHC) is a highly polymorphic genomic region that plays a central role in the immune system. We previously reported that only three MHC class II haplotypes (HP1-3) with one to three copies of MHC-IIA/IIB gene pairs (one copy of DAA/DAB locus and 0-2 copies of DBA/DBB loci) were detected among the five older founders, and four MHC-IIB exon 2 alleles (Type I-IV) were identified. In this study, MHC class II haplotypes in two novel founders, and MHC class IA genotypes at UAA locus in the seven founders were investigated. Of the two novel founders, while one possessed known HP1 and HP2, another possessed known HP1 and a novel haplotype (HP4) with the combination of type II and type I in DAB and DBB exon 2 s, respectively. Analysis of the linkage between MHC class II haplotypes and UAA alleles revealed five distinct MHC haplotypes against seven founders. These results strongly suggested that the founders might be considerably closely related, and the novel HP4 was produced by recombination between HP1 and HP2.

PubMedHuman reproduction open2026-07-11

Predicting natural conception leading to live birth for couples with infertility: a single-centre population-based cohort study of 7086 couples.

Cameron Natalie J NJ, Brian Kate K, McLernon David J DJ, Bhattacharya Siladitya S

Can a model be developed to predict natural conception leading to live birth over a period of 12 months in couples with different causes of infertility? We developed and validated a novel clinical prediction model that can be used to provide individualized estimates of the chance of a natural conception (leading to live birth) over a 12-month period for couples with different causes of infertility, including tubal factor, anovulation, male factor, unexplained, other (cervical, uterine, or sexual factor), and endometriosis. Existing prediction models for natural conception are primarily aimed at infertile couples with no identified cause (unexplained), mild male factor, or minimal endometriosis. Currently, there is no available model that is applicable across a wide range of fertility diagnoses at the point of initial assessment. A population-based cohort study based on data from a single large tertiary UK fertility centre serving the entirety of the North of Scotland, including all 9757 couples who registered at the clinic for the first time from 1998 to 2015. Using a Cox proportional hazards survival model, we estimated the chance of conception within the first year from diagnosis of infertility leading to live birth. The predictive accuracy of the model was assessed using discrimination and calibration measures in an internal validation. The clinical utility of the model was assessed using decision curve analysis. After exclusions, 7086 couples with infertility were included, of whom 891 (13%) had a natural conception within 1 year of diagnosis leading to live birth. Longer duration of infertility [hazard ratio (HR): 0.64 (95% CI: 0.57-0.72)], increasing female age [0.62 (0.55-0.70)], and tubal infertility [0.62 (0.47-0.81)] had the strongest influence on reducing the chance of natural conception within 1 year leading to live birth. Conversely, previous pregnancy [1.30 (1.12-1.50)] and unexplained infertility [1.29 (1.00-1.67)] were most strongly associated with increased chances of live birth. For example, a 25-year-old woman with 1 year of secondary unexplained infertility has a 33.8% predicted chance of having a baby resulting from natural conception within a year of diagnosis. In contrast, a 35-year-old woman with tubal infertility and 1 year of primary infertility has an estimated 6.0% predicted chance of live birth over a similar time horizon. The model demonstrated acceptable discrimination (optimism-corrected C-statistic 0.645) and good calibration in internal validation. Decision curve analysis demonstrated that applying the model at a 20% probability threshold would correctly identify an additional 7.2 couples per 100 as being likely to benefit from fertility treatment when compared against a 'treat-all' policy, which incorrectly assumes that all couples would benefit from fertility treatment. A freely available online calculator was constructed from the model formula to generate individual estimates of the chance of live birth following natural conception. The data used to inform this model were collected from a single centre until 2016, limiting generalizability. Any information not collected in this dataset, such as markers of ovarian reserve, severity of endometriosis, or subtype of ovulatory disorder, could not be included and may have improved the accuracy of the model predictions. As we have demonstrated that couples diagnosed with infertility can conceive on their own, knowledge of their individual chances of having a baby can clarify the net value of active treatment, including assisted reproduction. Use of this model via the online calculator could improve the quality of decision-making around the nature and timing of initiating fertility treatment. This work was funded in part by an NHS Grampian Charities Small Research Grant awarded to N.J.C, grant number SRG 24-30. We acknowledge the associated financial support of NHS Research Scotland, through NHS Grampian investment in the Grampian DaSH. N.J.C has no conflict of interest to declare. K.B. declares a previous role as Founder of the Fertility Alliance (charity) and receipt of speaker fees/honoraria from Merck and IBSA (paid to the Fertility Alliance). D.J.M. reports consulting fees from the Society for Assisted Reproductive Technology (SART) (paid to institution), honoraria from Merck for a fertility prediction modelling workshop, and financial support from ESHRE, Merck and IVIRMA to present at scientific conferences. S.B. reports royalties/licenses from Cambridge University Press, consulting fees from Merck, Ferring and Organon (paid to S.B. and to the institution), speaker fees/honoraria from Merck (paid to S.B. and to the institution), support for attending meetings/travel from Merck, and a leadership role as Board Member of the Fertility Alliance (charity). N/A.

PubMedHuman reproduction (Oxford, England)2026-07-08

ESHRE position paper: international limits on the number of offspring per gamete donor.

Frith Lucy L, Tassot Johanna J, Ahlstrom Aisling A, Baldani Dinka Pavičić DP et al.

How should the number of offspring per gamete donor be regulated at an international level? The European Society of Human Reproduction and Embryology (ESHRE) recommends introducing a European Union (EU)-wide limit on the number of families per gamete donor, starting at 50 families and gradually reducing it to a maximum of 15 families or lower, supported by an EU-wide donor registry to monitor compliance. Most European countries impose national limits on the number of offspring or families per donor, but these limits vary widely and are not always enforced. Cross-border movement of patients and the export of donor gametes between countries mean that large donor sibling groups can still emerge despite these restrictions. What matters to donor-conceived people is the total number of donor siblings, regardless of which country they are in, making a transnational limit the only relevant mechanism that can address this issue. This position paper sets out principles relevant to international donor offspring limits and the position and policy recommendations of ESHRE, focusing on the EU level. This ESHRE position paper was developed by a multidisciplinary expert working group. Recommendations are supported by data from the literature, where available. The first version was published for stakeholder review in November 2025, with 45 completed review forms received from organizations representing donor-conceived people, families built through donor conception and infertility patients, national fertility societies, researchers, professionals from different disciplines, and gamete banks. The paper was then revised on the basis of the stakeholder review. ESHRE considers that the wellbeing of donor-conceived people should have the highest priority when determining limits, while also balancing the wellbeing of prospective parents. Limits should be set for the number of families rather than individual children. ESHRE proposes a phased introduction starting at 50 families per donor, being reduced to a maximum of 15 families or lower, alongside a 20-year cap on distributing gametes to new families after the first donation. National limits should still be upheld where they are lower, and donors should be able to set their own lower personal limit. Compliance should be monitored through an EU-wide donor registry or, failing that, national registries, with gamete banks (including non-EU banks exporting into the EU) obliged to enforce the limit, donors required to declare all previous donations, and families counted as potential live births unless confirmed otherwise. The evidence base on the psychosocial impact of large donor sibling groups is small and developing, and definitive evidence of harm is limited. Research on the preferences of donor-conceived people, donors, and recipients regarding offspring limits is scarce and inconclusive. These recommendations therefore take a precautionary approach, and the proposed 15-family limit should be reviewed in light of developing knowledge during the transition period. An EU-wide limit would represent a feasible first step towards an international limit. An EU-wide donor registry could potentially serve secondary purposes such as supporting tracing in case of the diagnosis of a serious genetic condition and giving access to information to donors and donor-conceived people. Support for the working group was provided by ESHRE. L.F. and C.C.-J. report travel support from ESHRE. D.P.B. reports speakers' fees from Merck, Ferring, Gedeon Richter and MSD, travel support from ESHRE, and a position as the president of the Croatian Society for Gynaecological Endocrinology and Human Reproduction. A.A. reports speakers' fees from Merck Healthcare KGaA and Ferring, travel support from ESHRE, passive shareholder interest in Inception Midco 1. S.à r.l., membership in a subgroup of the European Medical Devices Coordination Group, and a position as vice chair of the EXPAMED panel on obstetrics, gynaecology and reproductive medicine. G.N. reports speakers' fees from Gedeon-Richter and Organon, travel support from ESHRE, and a position as past chairman and member of the Executive Committee of the Bulgarian Association for Human Reproductive Embryology. P.T. reports speakers' fees and travel support from Ferring and Gedeon Richter and a position as a board member on the Arbeitskreis donogene Insemination. J.K.-B. reports speakers' fees from Ferring, IBSA, Merck and CooperSurgical, travel support from Merck and ESHRE, an associate editor position for the journal Andrology, and a position as chair of the scientific advisory committee of the Association for Reproductive and Clinical Scientists (ARCS). The remaining authors (J.T. and N.V.) have nothing to declare. n/a.

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