Drug Database
LE

leuprolide acetate (Leupronax)

✓ Approved

Nanox · GNRH1 · Small Molecule

What is leuprolide acetate?

leuprolide acetate is a small molecule developed by Nanox. It is approved for therapeutic indications via injectable (others) or intramuscular (im) injection.

Drug Profile

Brand NamesLeupronax
CompanyNanox
Drug ClassSmall Molecule, Polypeptide
Molecular TargetGNRH1
RouteInjectable (Others), Intramuscular (IM) Injection
StatusApproved

Mechanism of Action

Molecular Targets

leuprolide acetate acts on 1 molecular target:

GNRH1gonadotropin releasing hormone 1 (GNRH, LHRH)
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Therapeutic Indications

leuprolide acetate is developed for 4 unique indications across 2 therapeutic areas.

Therapeutic AreaConditionPhase
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Breast cancer✓ Approved
Reproductive system and breast disordersEndometriosis✓ Approved
Neoplasms benign, malignant and unspecified (incl cysts and polyps)Prostate cancer✓ Approved
Reproductive system and breast disordersUterine fibrosis✓ Approved

Related Research Articles

PubMedJournal for immunotherapy of cancer2026-07-17

Blautia coccoides-derived acetate potentiates anti-PD-1 immunotherapy in melanoma by activating cytotoxic CD8+ T cells.

Zhang Zhiwen Z, Liang Xiaofeng X, Tian Yuyang Y, Li Chengyi C et al.

Gut microbiota can modulate cancer immunotherapy and enhance the efficacy of programmed cell death protein 1 (PD-1) blockade in tumors, yet the responsible microbes and underlying mechanisms remain incompletely understood. Publicly available anti-PD-1-treated melanoma microbiome cohorts were reanalyzed. Causal validation was performed using oral Blautia coccoides (B. coccoides) supplementation in B16-F10 melanoma-bearing mice. Untargeted and targeted liquid chromatography-tandem mass spectrometry-based metabolomics, CD8+ T-cell depletion, receptor identification and binding analyses, and downstream transcriptomic and biochemical assays were used to identify the key metabolite and investigate its mechanism of action. We identified Blautia as enriched in melanoma patients responding to immune checkpoint inhibitors, with higher abundance associated with non-progression. In melanoma-bearing mice, oral B. coccoides suppressed tumor growth and increased intratumoral effector CD8+ T cells. Metabolomic profiling identified acetate as a prominent B. coccoides-associated metabolite. Acetate enhanced CD8+ T-cell effector function. CD8+ T-cell depletion largely abrogated the antitumor effects of both B. coccoides and acetate, supporting a central role for CD8+ T cells. Mechanistically, these findings support a model in which acetate is associated with a TLR3-linked signaling pathway in CD8+ T cells, accompanied by PI3K/Akt activation and enhanced effector function. Notably, B. coccoides or acetate potentiated anti-PD-1 therapy in mouse melanoma models, supporting their potential as adjunctive strategies for melanoma immunotherapy. These findings support a model of an acetate-TLR3-linked PI3K/Akt signaling axis linking microbiota-associated metabolites to CD8+ T cell-mediated antitumor immunity. Importantly, our study highlights both B. coccoides and its derivative, acetate, as preclinical adjunctive candidates to potentiate anti-PD-1 efficacy in melanoma.

PubMedFrontiers in nutrition2026-07-17

Study on the migration regularity of volatile flavor compounds during the roasting process of Tartary buckwheat tea based on HS-GC-IMS and chemometrics.

Zhu Xianzhou X, Zhang Li L, Dai Zou Z, Guan Ju J et al.

Roasting is a critical processing step that strongly influences the chemical composition, volatile profile, and overall quality of Tartary buckwheat tea. This study investigated the dynamic changes in volatile flavor compounds during roasting using headspace-gas chromatography-ion mobility spectrometry (HS-GC-IMS) combined with chemometric analysis. Roasting significantly increased the contents of total flavonoids (2.29 g/100 g) and protein (15.67 g/100 g), while reducing the moisture content (5.77 g/100 g), particularly at stages X4-X6 (15-25 min). A total of 79 volatile compounds were identified by HS-GC-IMS, among which alcohols and ketones were predominant. Stages X3-X5 (10-20 min) were identified as the critical period for flavor accumulation. Partial least squares discriminant analysis (PLS-DA) identified 13 key discriminant compounds, including propyl acetate, hexyl butyrate, isoamyl formate, sec-butyl acetate, propanal, acrolein, 3-methyl-2-butenal, (E)-2-heptenal, methyl heptenone, 3-methyl-2-pentanone, 2-hexanone, sec-butanol, and 1-octene, as potential flavor markers. These findings clarify the roasting-dependent flavor evolution of Tartary buckwheat tea and provide a theoretical basis for process optimization to improve aroma quality.

PubMedACS applied materials & interfaces2026-07-17

Unveiling the Printability and Performance of 3D Printed Ethylene-Vinyl Acetate Stretchable Foams.

Rajabifar Nariman N, Ameli Amir A

The rise of additive manufacturing has pivoted the trajectory of advanced materials with intricate geometries and precise design. Although various materials have been adapted to 3D printing, developing printable microcellular foams remains in its infancy. Herein, for the first time, we report 3D printed ethylene-vinyl acetate (EVA) foams enabled by expandable microspheres (EMs). Expandable filaments of EVA/EMs containing 0-10 wt % EM result in a tailored density in the range of 0.903-0.224 g/cm3. The viable temperature spectrum relies upon EM content, where higher EM loading leads to a wider printing window. The foam density further exhibits an optimal correlation with temperature, reaching its minimum at 230 °C, independent of EM content. Microstructural analyses reveal uniform morphologies wherein the foam's cell density increases and cell size slightly drops with EM loading. The decay rate of Young's modulus and tensile strength with density reduction is significantly lower compared to conventional foams, which is attributed to the reinforcing effect of the EM shell material. Strain rate and print pattern dependency of mechanical properties are also discussed. While unfoamed EVA exhibits strain hardening upon cyclic compressive loading, the addition of EMs introduces a counteracting strain-softening behavior proportional to EM content. The thermal analysis furthermore depicts that EM leaves a negligible impact on the crystallinity of EVA. The findings of this work highlight the potential of 3D printed EVA foams as lightweight and tunable materials for various applications.

PubMedNature communications2026-07-17

Wavelength-dependent feedback behavior in light-gated polymersome nanoreactors.

Lathan Uthaya U, Kaya Beyzanur B, Matubbar Farzina F, Chami Mohamed M et al.

Biological systems integrate multiple feedback processes to regulate their adaptation to evolving stimuli with high specificity. Inspired by wavelength-selective feedback processes in visual signaling, we present a synthetic nanoreactor system capable of producing orthogonal, wavelength-dependent positive and negative feedback loops. Polymersomes functionalized with a broad-spectrum pyrazolone-based Donor-Acceptor Stenhouse Adduct (DASA) encapsulate an esterase enzyme and undergo light-gated permeability switching. Upon irradiation, the nanoreactors operate out-of-equilibrium, hydrolyzing ethyl acetate to generate acetic acid in a wavelength-programmed manner. Under yellow light (590 nm), positive feedback is mediated by spectral unmasking: acid-induced protonation of a solubilized dye decreases competition for yellow light, enhancing membrane permeability and enzyme activity, yielding a positive feedback loop. In contrast, blue light (405 nm) irradiation leads to the accumulation of the same dye that spectrally competes with the photoswitch, progressively suppressing membrane permeability by formation of a negative feedback loop. These stimulus-specific feedback dynamics enable reversible and tunable control over enzymatic reaction kinetics. Importantly, this platform introduces a paradigm shift for light-programmed, autonomous regulation in synthetic cell mimics and could open a pathway to dynamic modulation of microscale environments and biointerfaces without genetic intervention.

PubMedLangmuir : the ACS journal of surfaces and colloids2026-07-17

Dependence of Solvents and Surface Effects on Metal-Organic Framework Polymer Chain Interpenetration and Interfacial Stability.

Browe Matthew A MA, Hinkle Adam R AR, Iordanov Ivan O IO, Pearl Thomas P TP

Polymer-based coatings often incorporate fillers or inclusions into the polymer matrix to tune application-specific physical and chemical properties. Furthermore, the presence of specific solvents can either promote or impede dispersal of the inclusions and polymer chains. Here, all-atom molecular dynamics (MD) simulations are performed to probe the formation of interfacial regions in metal-organic framework (MOF)-polymer composites by including nanoscale crystallites of UiO-66 in a binder of a polyurethane or polyhydroxyurethane solvated with hexane or hexanol. We study the effect of different surface chemistries on the metal oxide nodes (hydroxyl, formate, or acetate groups), calculating polymer and solvent densities and interaction energies. We report secondary trends in chain adsorption (depletion) near the MOF surface as a function of different surface chemistries, while the polymer-solvent and solvent-solvent interactions appear as the primary factors controlling the interfacial uniformity. The simulations show that chain penetration into the MOF can be either entirely impeded by the choice of the blending solvent or promoted by the particular surface functionalization. Energetic barriers from the MD are directly extracted to quantify chain interpenetration of the MOF and reveal that interpenetration is a stabilizing process during interface formation and strongly dependent upon solvent presence and surface chemistry.

PubMedFood & function2026-07-17

In vitro fermentation characteristics of licochalcone A and its regulatory effects on human gut microbiota via multi-omics analysis.

Asif Ali A, Ziying Zou Z, Chen Ting T, Ahmad Ali A et al.

Historically, bioactive flavonoids from plant foods have been important components of the human diet and play key roles in shaping gut microbiota composition and host metabolism. Licochalcone A (LCA), a chalcone-type flavonoid derived from licorice (Glycyrrhiza spp.), has gained attention for its potential interactions with gut microbial communities. In the present study, an in vitro fecal batch fermentation system using samples from six healthy volunteers was used to characterize LCA-induced changes in microbial composition and metabolism. LCA was rapidly metabolized by the intestinal microbiota within 48 h, with pronounced interindividual variability among donors, indicating active microbial transformation. LCA treatment altered microbial activity by modifying short-chain fatty acid profiles, including acetate, propionate, and butyrate. LCA significantly increased the relative abundance of beneficial bacteria, including Prevotella, Segatella, and Bacteroides, while decreasing the abundance of taxa such as Fusobacterium and Escherichia. Untargeted metabolomics of the fermented broth revealed that LCA reshaped the gut metabolome, enriching metabolites involved in tryptophan metabolism and pantothenate and coenzyme A biosynthesis. Several metabolites, including Romucosine, Mosin C, and lucidone B, were altered, suggesting changes in microbial metabolic activity. Overall, these findings demonstrate that LCA can reshape gut microbial composition and metabolism, providing a basis for future development of functional foods.

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